National Natural Science Foundation of ChinaNational Natural Science Foundation of China (NSFC) [21272085, 21472056]
机构署名：
本校为第一且通讯机构
院系归属：
化学学院
摘要：
An NH2CN-promoted convergent integration of three self-sorting domino sequences is described for the construction of 6-iodo-3-methylthioimidazo[1,2-a] pyridines from aryl methyl ketones and 2-aminopyridines. This strategy allows the construction of an imidazo[1,2-a] pyridine ring along with methylthiolation at C-3 and iodination at C-6. Preliminary mechanistic studies indicate that this process terminates at the iodination stage without K...
