期刊论文

Ding, Ming-Wu

英文

中国化学快报：英文版

1001-8417

2015

26

9

1158-1160

10.1016/j.cclet.2015.06.011

Acknowledgments We gratefully acknowledge financial support of this work by the National Natural Science Foundation of China （No. 21172085）, the Natural Science Foundation of Hubei Province （No. 2014CFB567） and the Open Foundation of Hubei Province Key Laboratory of Purification and Application of Plant Anti-cancer Active Ingredients.

本校为通讯机构

A new efficient synthesis of 2,5,6-trisubstituted oxazolo[5,4-d]pyrimidi-7(6H)-ones by consecutive aza-Wittig reaction was developed. The sequential three-component reaction of oxazolyliminophosphorane 4, isocyanates and amines produced 2,5,6-trisubstituted oxazolo[5,4-d]pyrimidi-7(6H)-ones 7 in good overall yields in the presence of catalyti...

2,5,6-trisubstituted oxazolo 的新有效合成[5,4-d ] 由连续 aza-Wittig 反应的 pyrimidi-7 (6H ) 被开发。oxazolyliminophosphorane 的顺序的三部件的反应 4， isocyanates 和胺生产了 2,5,6-trisubstituted oxazolo [5,4-d ] 7 面对 EtONa 的催化数量在好外套产出的 pyrimidi-7 (6H ) 。