Novel sulfonylurea derivatives containing five-membered heterocycle 3a - l and 4a - d were synthesized in good yields by the regioselective addition of aryl sulfonylisocyanates 1 to 5-amino-3-benzyl (aryl) thio-1, 2, 4-triazoles and its pyrazole analogues 2. The structures of all these compounds were evaluated by elemental analyses and 1H NMR spectroscopy. The preliminary biological tests showed that the products displaye...